ARTEMISINE (QINGHAOSU) DERIVATIVES, THEIR PREPARATION METHODS AND THEIR USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

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专利名称 ARTEMISINE (QINGHAOSU) DERIVATIVES, THEIR PREPARATION METHODS AND THEIR USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 申请号 EP20060705603 专利类型 EP 公开(公告)号 EP1845099(B1) 公开(授权)日 2012.10.24 申请(专利权)人 中国科学院上海药物研究所 发明(设计)人 LI, YING;ZUO, JIANPING;YANG, ZHONGSHUN;ZHOU, WENLIANG;SUI, YI;WANG, JUNXIA;ZHANG, YU;ZHOU, YU;WU, JINMING 主分类号 C07D493/18 IPC主分类号 C07D493/18;A61K31/335;A61P37/00;C07D311/00;C07D321/00;C07D323/00 专利有效期 ARTEMISINE (QINGHAOSU) DERIVATIVES, THEIR PREPARATION METHODS AND THEIR USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 至ARTEMISINE (QINGHAOSU) DERIVATIVES, THEIR PREPARATION METHODS AND THEIR USE, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 法律状态 说明书摘要 The invention provides a type of artemisinin derivatives having following structure I, its preparation method and use, as well as a pharmaceutical composition containing such artemisinin derivatives and its use. The arteminsinin derivatives of the present invention and their pharmaceutical composition containing the artemisinin derivatives. have immunosuppressive activities and can be used more safely. The composition which comprises the artemisinin derivatives can be formulated into long-term dosage forms such as tablet, pellet and the like, and have wider productive and use value.

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